• AMPK製品生物活性の比較
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AMPK 阻害剤 | 活性剤 (7)


製品コード 製品名 製品説明 文献中の引用 カスタマーフィードバック
S2697 A-769662 A-769662は0.8μMのEC50による強力な、可逆的なAMPを起動するプロテインキナーゼ(AMPK)活性剤で、3.2μMでIC50で脂肪酸合成を禁止します。
S1802 AICAR (Acadesine) AICAR (Acadesine)の蓄積のアカデシン結果(それはAMPの両方の活性化効果を模倣します) AMPKとAMPKKの上で。
S7306 Dorsomorphin (Compound C) 2HCl Dorsomorphin (Compound C) 2HCl is a potent, reversible, selective AMPK inhibitor with Ki of 109 nM, exhibiting no significant inhibition of several structurally related kinases including ZAPK, SYK, PKCθ, PKA, and JAK3.
S2542 Phenformin HCl Phenformin HCl is a hydrochloride salt of phenformin that is an anti-diabetic drug from the biguanide class.
S7317 WZ4003 WZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively, without significant inhibition on 139 other kinases.
S7840 Dorsomorphin (Compound C)
S7318 HTH-01-015 HTH-01-015 is a potent and selective NUAK1 inhibitor with IC50 of 100 nM, >100-fold selectivity over NUAK2.