COX

COX 阻害剤 (43)

水溶性

製品コード 製品名 製品説明 文献中の引用 カスタマーフィードバック
S1261 Celecoxib セレコキシブは、40nMのIC50による選択的なCOX-2阻害剤です。
S1255 Nepafenac Nepafenac is a non-steroidal anti-inflammatory agent.
S1638 Ibuprofen Ibuprofen は非ステロイド薬(NSAID)、COX-1とCOX-2 を抑制すると、IC50 がそれぞれ13 μM 、370 μMになる.
S1723 Indomethacin Indomethacin(Indocid, Indocin) is a non-steroidal anti-inflammatory compound commonly used to reduce fever, pain, stiffness, and swelling.
S2007 Sulindac Sulindac (Clinoril) is a non-steroidal anti-inflammatory agent of the arylalkanoic acid class.
S7889 Xanthohumol Xanthohumol, a prenylated chalcone from hop, inhibits COX-1 and COX-2 activity and shows chemopreventive effects. Phase 1.
S7889 Xanthohumol Xanthohumol, a prenylated chalcone from hop, inhibits COX-1 and COX-2 activity and shows chemopreventive effects. Phase 1.
S7889 Xanthohumol Xanthohumol, a prenylated chalcone from hop, inhibits COX-1 and COX-2 activity and shows chemopreventive effects. Phase 1.
S7889 Xanthohumol Xanthohumol, a prenylated chalcone from hop, inhibits COX-1 and COX-2 activity and shows chemopreventive effects. Phase 1.
S7889 Xanthohumol Xanthohumol, a prenylated chalcone from hop, inhibits COX-1 and COX-2 activity and shows chemopreventive effects. Phase 1.
S1734 Meloxicam Meloxicam (Mobic) is a nonsteroidal anti-inflammatory agent with analgesic and fever reducer effects.
S3043 Rofecoxib Rofecoxib is a COX-2 inhibitor with IC50 of 18 nM.
S4295 Meclofenamate Sodium Meclofenamate Sodium is a dual COX-1/COX-2 inhibitor with IC50 of 40 nM and 50 nM, respectively, used in the treatment of joint, muscular pain, arthritis and dysmenorrhea.
S4248 Bromfenac Sodium Bromfenac is a nonsteroidal anti-inflammatory drug (NSAID) that has anti-inflammatory activity which may block prostaglandin synthesis by inhibiting cyclooxygenase 1 and 2.
S1518 Ibuprofen Lysine Ibuprofen Lysine is a non-steroidal anti-inflammatory drug.
S1646 Ketorolac Ketorolacは非選択COX阻害剤、人間COX-1とCOX-2に作用する時、IC50がそれぞれ1.23 µM と3.50 µM になる。
S1903 Diclofenac Sodium Diclofenac Sodium is a non-selective COX inhibitor with IC50 of 60 and 220 nM for ovine COX-1 and -2, respectively.
S1328 Etodolac Etodolac is a COX inhibitor with an IC50 of 53.5 nM.
S1645 Ketoprofen Ketoprofen is a non-selective NSAID with IC50 of 0.5 μM and 2.33 μM for human recombinant COX-1 and COX-2, respectively.
S1626 Naproxen Sodium Naproxen Sodiumは非選択エポキシ合酵素阻害剤(COX)、COX-1とCOX-2に作用する時、IC50がそれぞれ2.2μg / mLと1.3μg / mLになる。
S1713 Piroxicam Piroxicam is a non-selective COX inhibitor with an IC50 of 6 mM.
S1960 Pranoprofen Pranoprofen is a PGE2 inhibitor with IC50 of 7.5 μM.
S2602 Acemetacin Acemetacin is a non-steroidal anti-inflammatory drug and a glycolic acid ester of indometacin that is a cyclooxygenase inhibitor.
S2577 Phenacetin Phenacetin is a non-opioid analgesic without anti-inflammatory properties.
S1959 Tolfenamic Acid Tolfenamic acid is a COX-2 inhibitor with IC50 of 0.2 μM.
S2040 Nimesulide Nimesulide is a relatively COX-2 selective inhibitor with IC50 of 26 μM.
S2108 Flunixin Meglumin Flunixin Meglumin is a potent inhibitor of the enzyme cyclooxygenase used as analgesic agent with anti-inflammatory and antipyretic activity.
S3017 Aspirin Aspirin is a salicylate drug, often used as an analgesic to relieve minor aches and pains, as an antipyretic to reduce fever, and as an anti-inflammatory medication.
S3023 Bufexamac ブフェキサマックは、8.9μMのEC50によるIFN-αの分泌のための酵素シクロオキシゲナーゼとHDAC6/HDAC10阻害剤です。
S3018 Niflumic acid Niflumic acid is an inhibitor of cyclooxygenase-2 used for joint and muscular pain.
S4230 Oxaprozin Oxaprozin is a non-narcotic, non-steroidal anti-inflammatory drug (NSAID) used to relieve the inflammation, swelling, stiffness, and joint pain associated with osteoarthritis and rheumatoid arthritis.
S2047 Lornoxicam Lornoxicam is a COX-1 and COX-2 inhibitor with IC50 of 5 nM and 8 nM, respectively.
S3200 Triflusal Triflusal irreversibly inhibits the production of thromboxane-B2 in platelets by acetylating cycloxygenase-1.
S2903 Lumiracoxib Lumiracoxib is a novel, selective COX-2 inhibitor with IC50 and Ki of 0.14 μM and 0.06 μM, exhibits 515-fold selectivity over COX-1. Phase 4.
S3008 Zaltoprofen Zaltoprofen is an inhibitor of Cox-1 and Cox-2 for treatment of arthritis.
S4011 Ampiroxicam Ampiroxicamは、選択的でないシクロオキシゲナーゼ 抗炎症剤としての阻害剤です。
S4049 Valdecoxib Valdecoxibは、COX-2の強力で選択的な阻害体で、IC50が5 nMです。
S4051 Nabumetone Nabumetone is a non-steroidal anti-inflammatory drug and its active metabolite inhibits the COX.
S4078 Mefenamic Acid Mefenamic acidは、COX-1COX-2の競争的阻害体です。
S4136 Carprofen CarprofenはイヌCOX2を阻害、IC50 が 0.03 mMです。
S4149 Amfenac Sodium Monohydrate Amfenac Sodium monohydrate、酢酸部分を有する非ステロイド系鎮痛薬、抗炎症薬です。
S2531 Asaraldehyde Asaraldehyde is a selective COX-2 inhibitor.
S1761 Suprofen Suprofen(Profenal) is an NSAID.
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